denosumab


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denosumab

A monoclonal antibody drug that interferes with osteoclast production and function. The antibody binds to the receptor activator of a nuclear factor ligand RANKL, interfering with osteoclast differentiation, activation and survival. Given to post-menopausal women it increases bone mineral density and decreases the rate of bone reabsorption. The drug shows promise for the treatment of OSTEOPOROSIS.
Collins Dictionary of Medicine © Robert M. Youngson 2004, 2005
References in periodicals archive ?
Hsu et al., "An open-label, prospective pilot clinical study of denosumab for severe hyperparathyroidism in patients with low bone mass undergoing dialysis," The Journal of Clinical Endocrinology & Metabolism, vol.
Denosumab, a monoclonal antibody to the RANK ligand, has recently been used in a few cases and has been shown to decrease tumor burden size, reduce pain, resolve associated neurologic symptoms, and show evidence of radiographic healing [9-11].
Denosumab reduces bone resorption, increases bone mineral density (BMD), and reduces fracture risk [1].
Denosumab is a monoclonal antibody against the receptor activator of nuclear factor-[kappa][beta] ligand (RANKL), a cytokine that is essential for the formation, function, and survival of osteoclasts [6].
The patient subsequently began cycle 2 of cisplatin, doxorubicin, and cytoxan which was completed prior to discharge with a plan to initiate denosumab as an outpatient.
Denosumab is a human monoclonal antibody that inhibits normal and tumor associated RANKL [13-15].
More recently, RANK-Ligand inhibitors (denosumab) have also been used to reduce the risk of skeletal-related events in patients who have advanced cancers with bone metastases.
16 December 2015 - US-based biotechnology company Amgen (NASDAQ: AMGN) has entered into a definitive agreement with UK-based drugmaker GSK to reacquire all of its remaining rights to Prolia (denosumab), Xgeva (denosumab) and Vectibix (panitumumab) in 48 countries in Asia, South America, Europe, Australia and other regions throughout the world, the company said.
* 2 studies that explore the use of zoledronic acid or denosumab in women with breast cancer undergoing adjuvant therapy with an aromatase inhibitor
Denosumab is a fully-human, immunoglobulin G1 (IgG2) mAb against RANKL that is in Phase III of development for RA patients with active, erosive bone disease.
CHICAGO -- Postmenopausal women on denosumab for 8 years straight showed a continued nearlinear increase in bone mineral density at the lumbar spine as well as persistent reduction of bone turnover markers and a sustained low incidence of new vertebral and nonvertebral firactures in the ongoing FREEDOM open-label extension study.